SCHEMBL8809942

SCHEMBL8809942

COc1ccc2c(c1)c(OCCCN(C)C)nn2Cc1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.58
CYP1A2 P05177 2/20 0.58
HRH3 Q9Y5N1 2/20 0.58
GUCY1B2 O75343 1/20 0.58
CHRM2 P08172 1/20 0.58
HTR1A P08908 1/20 0.58
ADRA2A P08913 1/20 0.58
CYP2D6 P10635 1/20 0.58
CHRM1 P11229 1/20 0.58
DRD1 P21728 1/20 0.58
SLC6A2 P23975 1/20 0.58
SLC6A4 P31645 1/20 0.58
GUCY1A2 P33402 1/20 0.58
ADRA1A P35348 1/20 0.58
OPRM1 P35372 1/20 0.58
DRD3 P35462 1/20 0.58
SLC6A3 Q01959 1/20 0.58
GUCY1A1 Q02108 1/20 0.58
GUCY1B1 Q02153 1/20 0.58
KCNH2 Q12809 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978209 0.84 CNR1 (0.49) KDM4ECYP1A2HRH3GUCY1B2CHRM2
SCHEMBL8808522 0.84 KDM4E (0.82) KDM4ECYP1A2HRH3GUCY1B2CHRM2
SCHEMBL6974448 0.83 CNR1 (0.48) KDM4ECYP1A2HRH3GUCY1B2CHRM2
SCHEMBL6969602 0.79 CNR2 (0.52) KDM4ECNR2CNR1ACHE
SCHEMBL6969861 0.79 CNR2 (0.44) KDM4ECYP1A2HRH3GUCY1B2CHRM2
SCHEMBL6977954 0.78 CNR2 (0.53) KDM4ECYP1A2SLC6A4CNR2CNR1
SCHEMBL8809795 0.78 MET (0.50) KDM4ECYP1A2HRH3GUCY1B2CHRM2
SCHEMBL6966885 0.76 KDM4E (0.50) KDM4ECYP1A2HTR1APOLBCNR2
SCHEMBL9917395 0.76 HRH3 (0.77) KDM4ECYP1A2HRH3GUCY1B2CHRM2
SCHEMBL6968036 0.75 CNR1 (0.49) KDM4ECYP1A2POLBCNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775131-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA Medica Aktiengesellschaft (DE) 1997-05-28 EP disclosed
WO-1996004266-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1996-02-15 WO disclosed