SCHEMBL8809962

SCHEMBL8809962

CC(C)(C)OC(=O)NC(=O)C1(c2ccccc2)CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.51
HDAC1 Q13547 1/20 0.48
TACR1 P25103 1/20 0.47
TSHR P16473 2/20 0.45
ALOX15 P16050 1/20 0.45
ATM Q13315 1/20 0.45
HDAC4 P56524 2/20 0.42
ROCK2 O75116 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KHK P50053 1/20 0.39
ALDH1A1 P00352 1/20 0.39
THRB P10828 1/20 0.39
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AKT1 P31749 1/20 0.38
P2RX7 Q99572 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2273980 0.87 DRD2 (0.46) OPRM1HDAC4L3MBTL1ALDH1A1SMN1; SMN2
SCHEMBL8809179 0.87 CYP17A1 (0.40) OPRM1HDAC1TACR1TSHRALOX15
SCHEMBL8808902 0.86 ITGA4 (0.47) OPRM1HDAC1TACR1TSHRALOX15
SCHEMBL8806582 0.86 HDAC1 (0.41) OPRM1HDAC1TACR1
SCHEMBL8808488 0.82 AKT1 (0.37) OPRM1ALDH1A1HTTAKT1
SCHEMBL3892253 0.80 OPRM1 (0.45) OPRM1HDAC1TACR1TSHRALOX15
SCHEMBL6216344 0.80 OPRM1 (0.55) OPRM1HDAC1TACR1TSHRALOX15
SCHEMBL15200870 0.79 OPRM1 (0.54) OPRM1HDAC1TACR1HDAC4ROCK2
Hydrochloric Acid SCHEMBL27552695 0.78 OPRM1 (0.44) OPRM1HDAC1TACR1TSHRALOX15
SCHEMBL6544545 0.77 OPRM1 (0.57) OPRM1HDAC1TACR1HDAC4ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696280-B1 SUBSTITUTED PYRROLIDIN-3-YL-ALKYL-PIPERIDINES USEFUL AS TACHYKININ ANTAGONISTS MERRELL PHARMA INC (US) 1997-09-24 EP disclosed