SCHEMBL8810690

SCHEMBL8810690

Cc1cc(C)c(NC(=O)N(Cc2ccc(-c3ccsc3)cc2)C2CCCCCC2)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
BCL9 O00512 2/20 0.41
CTNNB1 P35222 2/20 0.41
POLB P06746 1/20 0.39
TP53 P04637 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HRH4 Q9H3N8 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
UBE2M P61081 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37
KMT2A Q03164 1/20 0.37
CCR5 P51681 3/20 0.37
MAPT P10636 1/20 0.37
KCNH2 Q12809 1/20 0.37
ROCK2 O75116 1/20 0.36
S1PR4 O95977 1/20 0.36
GCGR P47871 1/20 0.36
GIPR P48546 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809779 0.89 GAA (0.52) GAANPSR1POLBTP53ALDH1A1
SCHEMBL9056936 0.87 GAA (0.50) GAANPSR1TP53ALDH1A1UBE2M
SCHEMBL8808422 0.86 TP53 (0.52) GAANPSR1POLBTP53ALDH1A1
SCHEMBL8817749 0.86 NPSR1 (0.49) GAANPSR1POLBTP53ALDH1A1
SCHEMBL8807180 0.86 GAA (0.49) GAANPSR1TP53ALDH1A1HRH4
SCHEMBL8809768 0.85 GAA (0.48) GAANPSR1POLBTP53ALDH1A1
SCHEMBL8808615 0.84 CTSD (0.43) BCL9CTNNB1POLBTP53ALDH1A1
SCHEMBL8809295 0.83 ALDH1A1 (0.46) GAANPSR1BCL9CTNNB1ALDH1A1
SCHEMBL8806837 0.82 GAA (0.45) GAANPSR1TP53ALDH1A1HRH4
SCHEMBL8808845 0.81 GAA (0.51) GAANPSR1TP53ALDH1A1UBE2M

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784612-A1 UREA DERIVATIVES AND THEIR USE AS ACAT-INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-07-23 EP disclosed
WO-1996010559-A1 UREA DERIVATIVES AND THEIR USE AS ACAT-INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-04-11 WO disclosed