SCHEMBL8811089

SCHEMBL8811089

c1ccc2c(c1)CCC1(CCCNC1)S2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.46
HTR2C P28335 3/20 0.46
SIGMAR1 Q99720 3/20 0.46
HTR2B P41595 1/20 0.46
TMEM97 Q5BJF2 1/20 0.46
DRD2 P14416 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
CYP3A4 P08684 4/20 0.33
ALDH1A1 P00352 4/20 0.33
CYP2D6 P10635 4/20 0.33
USP2 O75604 3/20 0.33
CYP1A2 P05177 2/20 0.33
RYR2 Q92736 1/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8812960 0.72 HTR2A (0.34) HTR2AHTR2CSIGMAR1HTR2BCYP3A4
SCHEMBL24282934 0.68 HTR2C (0.39) HTR2AHTR2CSIGMAR1HTR2BTMEM97
SCHEMBL31059131 0.66 HTR2A (0.54) HTR2AHTR2CSIGMAR1HTR2BDRD2
SCHEMBL4882972 0.66 HTR2A (0.54) HTR2AHTR2CSIGMAR1HTR2BDRD2
SCHEMBL3169552 0.65 SIGMAR1 (0.44) HTR2AHTR2CSIGMAR1HTR2BTMEM97
SCHEMBL11285930 0.64 SIGMAR1 (0.42) HTR2AHTR2CSIGMAR1HTR2BTMEM97
SCHEMBL1222161 0.64 HTR2A (0.51) HTR2AHTR2CDRD2SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL27492472 0.64 SIGMAR1 (0.43) HTR2AHTR2CSIGMAR1HTR2BTMEM97
SCHEMBL9196136 0.64 HTR2A (0.81) HTR2AHTR2CDRD2SLC6A2SLC6A4
SCHEMBL7678355 0.62 SIGMAR1 (0.42) HTR2AHTR2CSIGMAR1HTR2BTMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997011697-A1 3-SPIROLACTAM, 3-SPIROAMINO, 3-SPIROLACTONE AND 3-SPIROBENZOPYRAN PIPERIDINES AND PYRROLIDINES PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1997-04-03 WO disclosed