SCHEMBL8811282

SCHEMBL8811282

O=C1NC(Cc2cccc3c2ccn3Cc2ccc(O)cc2)C(=O)S1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
HTR6 P50406 3/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.34
DBH P09172 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
BLM P54132 1/20 0.34
MPO P05164 1/20 0.33
SYK P43405 1/20 0.33
APP P05067 1/20 0.33
DNTT P04053 1/20 0.32
BACE1 P56817 1/20 0.32
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8812580 0.90 TNF (0.37) HTR6POLBMPOPARP1
SCHEMBL8685833 0.90 HTR6 (0.43) CHRNB2CHRNA7CHRNA4HTR6ALDH1A1
SCHEMBL8814121 0.89 PARP1 (0.41) HTR6CYP1A2CYP3A4TSHRMPO
SCHEMBL8811933 0.89 HTR6 (0.41) HTR6MPOPARP1
SCHEMBL8810754 0.89 PARP1 (0.41) HTR6ALDH1A1POLBCYP3A4MPO
SCHEMBL8811969 0.89 RHEB (0.40) HTR6MPOGAA
SCHEMBL8810209 0.87 CYP19A1 (0.40) POLBAPP
SCHEMBL8810917 0.87 CHRNB2 (0.41) CHRNB2CHRNA7CHRNA4HTR6POLB
SCHEMBL8813445 0.87 HTR6 (0.40) HTR6ALDH1A1CYP1A2CYP3A4MPO
Dimethylamine SCHEMBL8812830 0.86 HTR6 (0.43) CHRNB2CHRNA7CHRNA4HTR6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780389-A1 Thiazolidinedione derivatives, process for their preparation and pharmaceutical compositions containing them TOBISHI PHARMACEUTICAL CO., LTD. (JP) 1997-06-25 EP disclosed