SCHEMBL8813871

SCHEMBL8813871

CCC(C(N)=O)c1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.44
KCNQ2 O43526 1/20 0.41
ROCK1 Q13464 1/20 0.40
MYLK4 Q86YV6 1/20 0.40
BCL2L1 Q07817 1/20 0.40
BAD Q92934 1/20 0.40
CYP17A1 P05093 1/20 0.40
SCN9A Q15858 2/20 0.39
EPHX1 P07099 1/20 0.39
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5910306 0.95 KCNQ2 (0.44) KCNQ2EPHX1
SCHEMBL8813089 0.84 AKR1C3 (0.52) FFAR1BCL2L1BADAKR1C3AKR1C2
SCHEMBL23003724 0.81 KCNQ2 (0.47) KCNQ2
SCHEMBL27658097 0.81 ALDH1A1 (0.45) EPHX1
SCHEMBL15434306 0.78 EPHX1 (0.43) SCN9AEPHX1
SCHEMBL26898446 0.78 ALDH1A1 (0.50) EPHX1
SCHEMBL28234925 0.78 CRHBP (0.53) EPHX1
SCHEMBL4943215 0.78 LMNA (0.54) EPHX1
SCHEMBL9587806 0.78 KCNQ2 (0.45) KCNQ2
SCHEMBL15434362 0.78 EPHX1 (0.43) SCN9AEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684152-A CARBOXY DERIVATIVES FOR TREATMENT OF CARDIOVASCULAR DISORDERS MERCK & CO., INC. (US) 1997-11-04 US disclosed
WO-1997011936-A1 PREPARATION OF CARBOXYALKYL DERIVATIVES MERCK & CO., INC. (US) 1997-04-03 WO disclosed