SCHEMBL8815416

SCHEMBL8815416

COc1ccc(C)cc1-c1nc(-c2cccc(C)n2)nc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
ADORA2A P29274 1/20 0.44
TGFBR1 P36897 12/20 0.44
MAPK14 Q16539 1/20 0.44
ABCB1 P08183 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
ACACA Q13085 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8815721 0.90 KDM4E (0.53) KMT2AMEN1ADORA2ATGFBR1MAPK14
SCHEMBL8818491 0.89 IGF1R (0.43) KMT2AMEN1ADORA2ATGFBR1MAPK14
SCHEMBL8816854 0.89 ADORA2A (0.45) KMT2AMEN1ADORA2ATGFBR1MAPK14
SCHEMBL8816582 0.88 ADORA2A (0.58) KMT2AMEN1ADORA2ATGFBR1MAPK14
SCHEMBL8817891 0.85 TGFBR1 (0.47) KMT2AADORA2ATGFBR1MAPK14ALDH1A1
SCHEMBL8818706 0.83 TGFBR1 (0.46) ADORA2ATGFBR1MAPK14LMNA
SCHEMBL8817338 0.83 TGFBR1 (0.47) ADORA2ATGFBR1MAPK14LMNACYP1A2
SCHEMBL8818148 0.83 MEN1 (0.50) KMT2AMEN1ADORA2ATGFBR1MAPK14
SCHEMBL8818694 0.82 ADORA2A (0.48) KMT2AMEN1ADORA2ATGFBR1MAPK14
SCHEMBL8818335 0.82 L3MBTL1 (0.53) ABCB1ABCG2ACACAALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012066122-A1 2 - (PYRIDIN- 2 -YL) -QUINAZOLINE DERIVATIVES AND THEIR USE AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-24 WO disclosed