SCHEMBL8819232

SCHEMBL8819232

Cc1cccc(-c2nc(-c3ccc4c(c3)OCCCO4)c3ccccc3n2)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 6/20 0.55
MAPK14 Q16539 3/20 0.44
RIPK2 O43353 1/20 0.44
ACVR1B P36896 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CYP1A2 P05177 7/20 0.44
CYP3A4 P08684 7/20 0.44
CYP2D6 P10635 7/20 0.44
CYP2C19 P33261 6/20 0.44
USP2 O75604 5/20 0.44
HSD17B10 Q99714 5/20 0.44
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
CLK4 Q9HAZ1 4/20 0.44
ALOX15 P16050 4/20 0.44
MAPK1 P28482 4/20 0.44
LMNA P02545 3/20 0.44
TSHR P16473 3/20 0.44
CYP2C9 P11712 2/20 0.44
ALDH1A1 P00352 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8816383 0.91 TGFBR1 (0.66) TGFBR1MAPK14RIPK2ACVR1BTDP1
SCHEMBL8818164 0.87 TGFBR1 (0.50) TGFBR1MAPK14RIPK2ACVR1BTDP1
SCHEMBL8815687 0.80 TGFBR1 (0.49) TGFBR1MAPK14CYP1A2MEN1KMT2A
SCHEMBL8819429 0.79 TGFBR1 (0.48) TGFBR1MAPK14MEN1KMT2A
SCHEMBL6120916 0.78 TGFBR1 (0.54) TGFBR1MAPK14MEN1KMT2AALDH1A1
SCHEMBL8814729 0.78 NR1I3 (0.54) TGFBR1MAPK14MEN1KMT2ALMNA
SCHEMBL8817137 0.77 TGFBR1 (0.54) TGFBR1MAPK14MEN1KMT2AALDH1A1
SCHEMBL8816391 0.77 ALDH1A1 (0.56) TGFBR1MAPK14TDP1CYP1A2MEN1
SCHEMBL8818425 0.77 TGFBR1 (0.46) TGFBR1MAPK14LMNAALDH1A1KDM4E
SCHEMBL8816897 0.77 TGFBR1 (0.46) TGFBR1MAPK14MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012066122-A1 2 - (PYRIDIN- 2 -YL) -QUINAZOLINE DERIVATIVES AND THEIR USE AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-24 WO disclosed