SCHEMBL8819877

SCHEMBL8819877

CC(=O)Oc1ccc(OCc2ccccc2)c(N(C(=O)OC(C)(C)C)S(=O)(=O)c2cccc3ccccc23)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 5/20 0.40
NFE2L2 Q16236 4/20 0.40
HTR6 P50406 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MTNR1A P48039 2/20 0.35
MTNR1B P49286 2/20 0.35
NR1D1 P20393 1/20 0.35
PTPN1 P18031 1/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP19A1 P11511 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8817183 0.88 NQO2 (0.40) KEAP1NFE2L2MRGPRX4NPSR1NPC1
SCHEMBL3286247 0.87 KEAP1 (0.43) KEAP1NFE2L2PTPN1MEN1POLB
SCHEMBL6140114 0.81 AR (0.39) NPC1RAB9ASMN1; SMN2L3MBTL1MTNR1A
SCHEMBL6139688 0.76 CYP19A1 (0.45) KEAP1NFE2L2MAPTSMN1; SMN2L3MBTL1
SCHEMBL3287375 0.75 KEAP1 (0.42) KEAP1NFE2L2NPSR1MAPTSMN1; SMN2
SCHEMBL7467733 0.73 CYP19A1 (0.44) MAPTSMN1; SMN2L3MBTL1CYP19A1
SCHEMBL5264076 0.72 KEAP1 (0.40) KEAP1NFE2L2MEN1KMT2A
SCHEMBL3289538 0.72 KEAP1 (0.40) KEAP1NFE2L2MEN1KMT2A
SCHEMBL3142761 0.71 MEN1 (0.40) MAPTSMN1; SMN2MEN1KMT2ACYP19A1
SCHEMBL5203422 0.71 MEN1 (0.40) MAPTSMN1; SMN2MEN1KMT2ACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997034905-A1 PHOSPHORUS CONTAINING ARYLOXY AND ARYLTHIOPROPANOL AMINE DERIVATIVES USEFUL AS BETA ADRENORECEPTOR AGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-09-25 WO disclosed