SCHEMBL8828181

SCHEMBL8828181

COc1ccc(CCN(C)CCCN(C)C(=O)/C=C/c2ccc(F)cc2)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.52
CYP2D6 P10635 2/20 0.52
CYP1A2 P05177 1/20 0.52
BLM P54132 1/20 0.51
PMP22 Q01453 1/20 0.51
MMP1 P03956 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
CYP2C9 P11712 3/20 0.49
CYP2C19 P33261 3/20 0.49
SMPD1 P17405 1/20 0.49
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 2/20 0.47
MAPT P10636 4/20 0.47
ABCB1 P08183 1/20 0.47
APP P05067 1/20 0.46
KCNH2 Q12809 1/20 0.45
IKBKB O14920 1/20 0.45
CHUK O15111 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828421 0.92 CYP3A4 (0.56) CYP3A4CYP2D6CYP1A2BLMPMP22
SCHEMBL8828304 0.89 SMPD1 (0.49) CYP3A4CYP2D6CYP1A2BLMPMP22
SCHEMBL8828198 0.89 APP (0.51) CYP3A4CYP2D6CYP1A2BLMPMP22
SCHEMBL8828234 0.86 CYP3A4 (0.50) CYP3A4CYP2D6CYP1A2BLMPMP22
SCHEMBL8828259 0.84 MAPT (0.62) MEN1KMT2AALDH1A1KDM4ELMNA
SCHEMBL4878047 0.83 APP (0.62) CYP3A4CYP2D6CYP1A2BLMPMP22
SCHEMBL4878055 0.83 APP (0.62) CYP3A4CYP2D6CYP1A2BLMPMP22
SCHEMBL8828400 0.80 CYP3A4 (0.47) CYP3A4CYP2D6CYP1A2BLMPMP22
SCHEMBL8828237 0.80 APP (0.51) CYP3A4CYP2D6CYP1A2BLMPMP22
SCHEMBL8828274 0.79 OPRM1 (0.49) CYP3A4CYP2D6CYP1A2BLMPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684163-A Process for the preparation of N-(ortho-alkylphenyl)-imides BAYER AKTIENGESELLSCHAFT (DE) 1997-11-04 US disclosed
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed