SCHEMBL8828274

SCHEMBL8828274

COc1ccc(CCN(C)CCCNC(=O)C/C=C/c2ccc(F)cc2)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.49
TMEM97 Q5BJF2 2/20 0.49
SIGMAR1 Q99720 2/20 0.49
CYP3A4 P08684 5/20 0.48
CYP2D6 P10635 2/20 0.48
CYP1A2 P05177 1/20 0.48
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
ALDH1A1 P00352 4/20 0.47
CYP2C9 P11712 3/20 0.46
CYP2C19 P33261 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 4/20 0.46
KDM4E B2RXH2 1/20 0.45
OPRK1 P41145 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8828196 0.99 BLM (0.49) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6
SCHEMBL8828131 0.92 CYP3A4 (0.52) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6
SCHEMBL8828235 0.92 MAPT (0.56) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6
SCHEMBL8828147 0.92 MAPT (0.56) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6
SCHEMBL8828272 0.91 OPRM1 (0.47) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6
SCHEMBL8828252 0.91 MAPT (0.49) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6
SCHEMBL8828188 0.91 LMNA (0.49) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6
SCHEMBL8828425 0.91 MEN1 (0.41) OPRM1TMEM97SIGMAR1ALDH1A1MEN1
SCHEMBL8828550 0.90 OPRM1 (0.49) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6
SCHEMBL8828423 0.90 MAPT (0.53) OPRM1TMEM97SIGMAR1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP claimed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US claimed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP claimed
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed