SCHEMBL8828320

SCHEMBL8828320

O=C(O)C/C=C/c1ccc(Cl)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PAM P19021 1/20 0.56
GRIK1 P39086 1/20 0.54
GRIK2 Q13002 1/20 0.54
PYGL P06737 11/20 0.53
ALDH1A1 P00352 1/20 0.47
GUSB P08236 1/20 0.44
GPR183 P32249 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
PTGS2 P35354 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828326 1.00 PAM (0.56) PAMGRIK1GRIK2PYGLALDH1A1
SCHEMBL28564125 0.85 PAM (0.51) PAMGRIK1GRIK2PYGLALDH1A1
SCHEMBL8063786 0.83 GRIK1 (0.51) GRIK1GRIK2PYGLALDH1A1GUSB
SCHEMBL9492222 0.80 PYGL (0.46) GRIK1GRIK2PYGLALDH1A1GUSB
SCHEMBL9046738 0.79 PAM (0.68) PAMGRIK1GRIK2ALDH1A1
SCHEMBL9046744 0.79 PAM (0.68) PAMGRIK1GRIK2ALDH1A1
Acetic Acid SCHEMBL6974964 0.79 GRIK1 (0.51) GRIK1GRIK2PYGLALDH1A1GUSB
SCHEMBL3743993 0.77 ALDH1A1 (0.57) GRIK1GRIK2PYGLALDH1A1GUSB
SCHEMBL2092421 0.77 ALDH1A1 (0.54) GRIK1GRIK2PYGLALDH1A1GUSB
SCHEMBL2092419 0.77 ALDH1A1 (0.54) GRIK1GRIK2PYGLALDH1A1GUSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed