SCHEMBL8828322

SCHEMBL8828322

COc1ccc(CCN(C)CCCNC(=O)C/C=C/c2cc(OC)c(OC)c(OC)c2)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
KDM4E B2RXH2 2/20 0.56
PKM P14618 1/20 0.56
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
OPRM1 P35372 3/20 0.49
TMEM97 Q5BJF2 3/20 0.49
SIGMAR1 Q99720 3/20 0.49
CYP3A4 P08684 3/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
PMP22 Q01453 2/20 0.48
BLM P54132 1/20 0.48
OPRK1 P41145 2/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
CACNA1F O60840 1/20 0.45
LMNA P02545 1/20 0.45
ABCB1 P08183 1/20 0.45
HTR1A P08908 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828131 0.93 CYP3A4 (0.52) ALDH1A1KDM4EMEN1KMT2AOPRM1
SCHEMBL8828235 0.89 MAPT (0.56) ALDH1A1KDM4EMEN1KMT2AOPRM1
SCHEMBL8828147 0.89 MAPT (0.56) ALDH1A1PKMMEN1KMT2AOPRM1
SCHEMBL8828252 0.88 MAPT (0.49) ALDH1A1KDM4EMEN1KMT2AOPRM1
SCHEMBL8828188 0.88 LMNA (0.49) ALDH1A1MEN1KMT2AOPRM1TMEM97
SCHEMBL8828274 0.88 OPRM1 (0.49) ALDH1A1KDM4EMEN1KMT2AOPRM1
SCHEMBL8828305 0.87 OPRM1 (0.47) ALDH1A1MEN1KMT2AOPRM1TMEM97
SCHEMBL8828362 0.87 LMNA (0.59) ALDH1A1MEN1KMT2AOPRM1TMEM97
SCHEMBL8828423 0.87 MAPT (0.53) ALDH1A1MEN1KMT2AOPRM1TMEM97
Hydrochloric Acid SCHEMBL8828196 0.87 BLM (0.49) ALDH1A1KDM4EMEN1KMT2AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed