SCHEMBL8828323

SCHEMBL8828323

O=C(O)C/C=C/c1ccccc1F

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PAM P19021 1/20 0.58
NFE2L2 Q16236 7/20 0.54
MAOB P27338 2/20 0.46
CYP1A2 P05177 3/20 0.44
CYP1B1 Q16678 2/20 0.44
CYP2D6 P10635 1/20 0.44
CYP1A1 P04798 1/20 0.43
MAPT P10636 2/20 0.43
RECQL P46063 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828328 1.00 PAM (0.58) PAMNFE2L2MAOBCYP1A2CYP1B1
SCHEMBL24536155 0.86 PAM (0.50) PAMNFE2L2CYP2D6
SCHEMBL27301670 0.83 PAM (0.47) PAMNFE2L2MAOBCYP2D6RAB9A
SCHEMBL30942501 0.83 PAM (0.47) PAMNFE2L2MAOBCYP2D6RAB9A
SCHEMBL27799088 0.79 PAM (0.60) PAMMAOBCYP2D6SMN1; SMN2
SCHEMBL9150858 0.79 PAM (0.60) PAMNFE2L2CYP1B1CYP1A1MAPT
SCHEMBL30443677 0.78 PAM (0.58) PAMMAOBCYP1A2CYP1B1CYP2D6
SCHEMBL15540625 0.78 PAM (0.58) PAMMAOBCYP1A2CYP1B1CYP2D6
SCHEMBL15540628 0.78 PAM (0.58) PAMMAOBCYP1A2CYP1B1CYP2D6
SCHEMBL28010950 0.78 PAM (0.58) PAMMAOBCYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed