SCHEMBL882833

SCHEMBL882833

CC(C)(C)OC(=O)N1C2CC2C[C@H]1c1ncc(-c2ccc(C#Cc3ccc4c(ccc5nc([C@@H]6CC7CC7N6C(=O)OC(C)(C)C)[nH]c54)c3)cc2)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 3/20 0.34
SSTR3 P32745 1/20 0.34
GABRA1 P14867 2/20 0.31
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
GABRA3 P34903 2/20 0.31
GABRA2 P47869 2/20 0.31
NR1I2 O75469 1/20 0.30
ABCB11 O95342 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
OPRK1 P41145 1/20 0.30
KCNH2 Q12809 1/20 0.30
PRCP P42785 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16229701 0.93 SSTR3 (0.35) HPGDSSSTR3
SCHEMBL12328003 0.92 HPGDS (0.36) HPGDSSSTR3NR1I2ABCB11CYP3A4
SCHEMBL16229709 0.91 GABRA1 (0.35) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL13221409 0.89 HPGDS (0.36) HPGDSSSTR3GABRA1GABRG2GABRB3
SCHEMBL10201173 0.89 HPGDS (0.36) HPGDSSSTR3GABRA1GABRG2GABRB3
SCHEMBL12373653 0.87 GABRA1 (0.35) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL10202474 0.87 GABRA1 (0.35) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL12295800 0.86 GABRA5 (0.38) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL883264 0.85 CYP3A4 (0.42) HPGDSNR1I2ABCB11CYP3A4CYP2C9
SCHEMBL12328180 0.85 KRAS (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012039717-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-29 WO disclosed
WO-2010117635-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-10-14 WO disclosed