SCHEMBL8828558

SCHEMBL8828558

CN(C)C(=O)c1cc(C#N)ccc1NCCCOS(C)(=O)=O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 1/20 0.38
NR3C1 P04150 1/20 0.37
CDK2 P24941 1/20 0.37
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
CDK19 Q9BWU1 1/20 0.36
CDK1 P06493 1/20 0.35
CXCR2 P25025 1/20 0.33
TBXA2R P21731 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
NCEH1 Q6PIU2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828665 0.80 ADRA1D (0.44) NR3C1CXCR2
SCHEMBL13943063 0.66 EGLN1 (0.40) CDK1CXCR2PDK1PDK2PDK3
SCHEMBL7191231 0.65 PTGER4 (0.48) KAT2B
SCHEMBL18398655 0.65 ADRA1D (0.47) CDK2CXCR2
SCHEMBL30033113 0.65 FLT1 (0.48) CDK2PDK1PDK2PDK3PDK4
SCHEMBL2903095 0.65 MAPT (0.51)
SCHEMBL7959199 0.65 ALDH1A1 (0.51)
SCHEMBL7179435 0.65 KAT2B (0.64) KAT2B
SCHEMBL18398613 0.65 ADRA1D (0.48) CDK2CXCR2
SCHEMBL6214912 0.64 KAT2B (0.45) KAT2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed