SCHEMBL8832369

SCHEMBL8832369

N=C(N)NC(=O)c1ccc(Oc2ccc3ncccc3c2)c(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.46
TRPM8 Q7Z2W7 6/20 0.44
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 2/20 0.41
SCN9A Q15858 2/20 0.41
ABL1 P00519 1/20 0.41
SRC P12931 1/20 0.41
ALOX15 P16050 1/20 0.41
HTT P42858 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
SCD O00767 1/20 0.39
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
BRAF P15056 1/20 0.39
PARG Q86W56 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8831746 0.82 PLK1 (0.47) PLK1NPC1RAB9AALDH1A1SCN9A
SCHEMBL8831863 0.81 SMN1; SMN2 (0.49) NPC1RAB9AALDH1A1ABL1GAA
Hydrochloric Acid SCHEMBL8379790 0.80 SMN1; SMN2 (0.48) NPC1RAB9AALDH1A1ABL1GAA
Hydrochloric Acid SCHEMBL8503960 0.79 STK39 (0.45) SCN9AHDAC1SMN1; SMN2
SCHEMBL8767698 0.79 F2 (0.45) SCN9AHDAC1HDAC2SMN1; SMN2BRAF
Hydrochloric Acid SCHEMBL8505884 0.78 F2 (0.44) SCN9AHDAC1HDAC2SMN1; SMN2BRAF
Hydrochloric Acid SCHEMBL8506593 0.77 BRAF (0.43) RAB9AHDAC1HDAC2BRAFPARG
SCHEMBL8070147 0.76 TSHR (0.40) ALDH1A1HTT
SCHEMBL8059411 0.75 HDAC3 (0.39) SCN9AHDAC1HDAC2BRAF
SCHEMBL8881133 0.75 PARG (0.35) SCN9AHDAC1HDAC2BRAFPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5665739-A CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-09-09 US disclosed