SCHEMBL8833233

SCHEMBL8833233

C=CCOC(=O)NCCCI

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 8/20 0.40
ERN1 O75460 3/20 0.39
HRH4 Q9H3N8 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
TGM2 P21980 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
EPHX2 P34913 1/20 0.36
TSHR P16473 1/20 0.36
MAPT P10636 1/20 0.36
CACNA1B Q00975 1/20 0.36
APBA1 Q02410 1/20 0.36
BRD4 O60885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21105283 0.89 MEN1 (0.38) ACHEERN1HRH4HRH3TGM2
SCHEMBL3676772 0.86 TGM2 (0.46) ACHEERN1TGM2EPHX2TSHR
SCHEMBL24660419 0.85 HRH4 (0.49) ACHEERN1HRH4HRH3TGM2
SCHEMBL13055388 0.84 MAPT (0.42) ACHEERN1HRH4HRH3MEN1
SCHEMBL15809690 0.83 ACHE (0.46) ACHEERN1HRH4HRH3TGM2
SCHEMBL4678545 0.83 ACHE (0.41) ACHEERN1HRH4HRH3TGM2
SCHEMBL8781903 0.82 MEN1 (0.39) ACHEERN1HRH4HRH3MEN1
SCHEMBL15109209 0.81 ALDH1A1 (0.46) ACHEERN1HRH4HRH3TGM2
SCHEMBL8769203 0.81 ACHE (0.63) ACHETSHR
SCHEMBL9547242 0.81 ERN1 (0.40) ACHEERN1HRH4HRH3TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5608056-A Substituted 3-pyrrolidinylthio-carbapenems as antimicrobial agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-04 US disclosed
EP-0636133-A1 SUBSTITUTED 3-PYRROLIDINYLTHIO-CARBAPENEMS AS ANTIMICROBIAL AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-02-01 EP disclosed
WO-1993021186-A1 SUBSTITUTED 3-PYRROLIDINYLTHIO-CARBAPENEMS AS ANTIMICROBIAL AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-10-28 WO disclosed