SCHEMBL8835575

SCHEMBL8835575

CCOC(=O)c1[nH]c2cc(Cl)cc(Cl)c2c1NCc1cccc(CC(=O)c2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 10/20 0.51
GRIN1 Q05586 3/20 0.45
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
HPGD P15428 1/20 0.43
XBP1 P17861 1/20 0.43
CYP2C19 P33261 1/20 0.43
TP53 P04637 1/20 0.42
MDM2 Q00987 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835392 0.88 GRIN1 (0.55) GRIN1CYP1A2
SCHEMBL8835573 0.87 ALOX15 (0.46) ALOX15GRIN1ALDH1A1CYP1A2HPGD
SCHEMBL4341047 0.85 ALDH1A1 (0.48) ALOX15GRIN1ALDH1A1CYP1A2HPGD
SCHEMBL8545149 0.83 ALDH1A1 (0.49) ALOX15GRIN1ALDH1A1CYP1A2HPGD
SCHEMBL8539658 0.81 ALDH1A1 (0.48) ALOX15GRIN1ALDH1A1CYP1A2HPGD
SCHEMBL8835577 0.79 ALOX15 (0.45) ALOX15GRIN1ALDH1A1CYP1A2HPGD
SCHEMBL8540435 0.79 TP53 (0.48) ALOX15ALDH1A1CYP1A2HPGDXBP1
SCHEMBL8538422 0.78 ALDH1A1 (0.44) ALOX15GRIN1ALDH1A1CYP1A2HPGD
SCHEMBL8835655 0.78 ALDH1A1 (0.48) ALOX15GRIN1ALDH1A1CYP1A2HPGD
SCHEMBL8543504 0.78 ALOX15 (0.47) ALOX15ALDH1A1CYP1A2HPGDXBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5703107-A CENTRAL NERVOUS SYSTEM DISORDERS; ANALGESICS; ANTIEPILEPTIC AGENTS MERRELL PHARMACEUTICALS INC. (US) 1997-12-30 US disclosed
US-5675018-A 3-amidoindolyl derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-10-07 US disclosed