SCHEMBL8835577

SCHEMBL8835577

CCOC(=O)c1[nH]c2cc(Cl)c(NCc3ccccc3)c(Cl)c2c1CC(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.45
HPGD P15428 2/20 0.44
KDM4E B2RXH2 1/20 0.44
GRIN1 Q05586 2/20 0.40
NPC1 O15118 1/20 0.40
CASP3 P42574 1/20 0.40
RAB9A P51151 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
MAPT P10636 1/20 0.40
MCL1 Q07820 1/20 0.40
HTR6 P50406 2/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
XBP1 P17861 1/20 0.39
CYP2C19 P33261 1/20 0.39
MDM2 Q00987 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835393 0.88 GRIN1 (0.53) KDM4EGRIN1MCL1
SCHEMBL8835832 0.80 HPGD (0.45) ALOX15HPGDKDM4ENPC1CASP3
SCHEMBL8835575 0.79 ALOX15 (0.51) ALOX15HPGDGRIN1TP53ALDH1A1
SCHEMBL8836023 0.77 MDM2 (0.44) HPGDKDM4ECASP3RAB9AMAPT
SCHEMBL8835573 0.75 ALOX15 (0.46) ALOX15HPGDKDM4EGRIN1LMNA
SCHEMBL8835837 0.73 ALDH1A1 (0.39) ALOX15HPGDKDM4ENPC1CASP3
SCHEMBL4341047 0.72 ALDH1A1 (0.48) ALOX15HPGDKDM4EGRIN1NPC1
SCHEMBL8541953 0.71 ALOX15 (0.48) ALOX15HPGDKDM4EMAPTTP53
SCHEMBL8545149 0.71 ALDH1A1 (0.49) ALOX15HPGDKDM4EGRIN1MAPT
SCHEMBL8542212 0.69 ALOX15 (0.48) ALOX15HPGDKDM4ERAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5703107-A CENTRAL NERVOUS SYSTEM DISORDERS; ANALGESICS; ANTIEPILEPTIC AGENTS MERRELL PHARMACEUTICALS INC. (US) 1997-12-30 US disclosed
US-5675018-A 3-amidoindolyl derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-10-07 US disclosed