Demannose

Demannose

SCHEMBL8835653

NO.O=C[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)CO

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
TDP1 Q9NUW8 1/20 0.50
USP2 O75604 1/20 0.45
SLCO1B1 Q9Y6L6 1/20 0.45
PDE4A P27815 1/20 0.43
AKR1B1 P15121 1/20 0.40
KDM4E B2RXH2 2/20 0.38
MPI P34949 1/20 0.33
CYP2C19 P33261 1/20 0.32
HIF1A Q16665 1/20 0.32
TOP1 P11387 1/20 0.32
PAX8 Q06710 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Demannose SCHEMBL27550245 1.00 LMNA (0.52) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL4303243 1.00 LMNA (0.52) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL11361073 0.95 LMNA (0.52) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL6529193 0.95 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL13947310 0.95 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL1812 0.95 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL525084 0.95 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL20500378 0.95 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL1051912 0.95 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
Demannose SCHEMBL2290731 0.95 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180284106-A1 METHOD OF QUANTIFYING PEPTIDE-DERIVATIVE LIBRARIES USING PHAGE DISPLAY 48Hour Discovery Inc. (CA) 2018-10-04 US claimed
US-20150024958-A1 METHOD OF QUANTIFYING PEPTIDE-DERIVATIVE LIBRARIES USING PHAGE DISPLAY THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2015-01-22 US claimed
EP-2810069-A1 METHOD OF QUANTIFYING PEPTIDE-DERIVATIVE LIBRARIES USING PHAGE DISPLAY The Governors of the University of Alberta (CA) 2014-12-10 EP claimed
WO-2013113127-A1 METHOD OF QUANTIFYING PEPTIDE-DERIVATIVE LIBRARIES USING PHAGE DISPLAY THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2013-08-08 WO claimed
EP-4350056-A2 GENETIC ENCODING OF CHEMICAL POST-TRANSLATIONAL MODIFICATION FOR PHAGE-DISPLAYED LIBRARIES The Governors Of The University Of Alberta (CA) 2024-04-10 EP disclosed
EP-3209819-B1 GENETIC ENCODING OF CHEMICAL POST-TRANSLATIONAL MODIFICATION FOR PHAGE-DISPLAYED LIBRARIES UNIV ALBERTA (CA) 2024-02-14 EP disclosed
US-10724034-B2 Genetic encoding of chemical post-translational modification for phage-displayed libraries 48Hour Discovery Inc. (CA) 2020-07-28 US disclosed
US-20180284106-A1 METHOD OF QUANTIFYING PEPTIDE-DERIVATIVE LIBRARIES USING PHAGE DISPLAY 48Hour Discovery Inc. (CA) 2018-10-04 US disclosed
US-9958437-B2 Method of quantifying peptide-derivative libraries using phage display THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2018-05-01 US disclosed
US-20170355982-A1 GENETIC ENCODING OF CHEMICAL POST-TRANSLATIONAL MODIFICATION FOR PHAGE-DISPLAYED LIBRARIES THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2017-12-14 US disclosed
EP-3209819-A1 GENETIC ENCODING OF CHEMICAL POST-TRANSLATIONAL MODIFICATION FOR PHAGE-DISPLAYED LIBRARIES The Governors Of The University Of Alberta (CA) 2017-08-30 EP disclosed
US-20150024958-A1 METHOD OF QUANTIFYING PEPTIDE-DERIVATIVE LIBRARIES USING PHAGE DISPLAY THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2015-01-22 US disclosed
EP-2810069-A1 METHOD OF QUANTIFYING PEPTIDE-DERIVATIVE LIBRARIES USING PHAGE DISPLAY The Governors of the University of Alberta (CA) 2014-12-10 EP disclosed
WO-2013113127-A1 METHOD OF QUANTIFYING PEPTIDE-DERIVATIVE LIBRARIES USING PHAGE DISPLAY THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2013-08-08 WO disclosed
US-5599988-A CONDENSATION, CYCLIZATION SMITHKLINE BEECHAM CORPORATION (US) 1997-02-04 US disclosed
WO-1996019438-A1 AN ENANTIOSELECTIVE SYNTHESIS OF CERTAIN HYDROXYLAMINES SMITHKLINE BEECHAM CORPORATION (US) 1996-06-27 WO disclosed