SCHEMBL8837787

SCHEMBL8837787

O=C(O)c1cccc(-c2ccnc(Nc3cccc(OC(F)(F)C(F)F)c3)n2)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 7/20 0.71
BCR P11274 7/20 0.71
PRKCA P17252 6/20 0.71
CSNK2A1 P68400 1/20 0.64
SRC P12931 4/20 0.60
PRKCD Q05655 3/20 0.60
EGFR P00533 2/20 0.60
PRKACA P17612 2/20 0.60
PRKACG P22612 2/20 0.60
PRKACB P22694 2/20 0.60
SYK P43405 5/20 0.59
MAPK8 P45983 1/20 0.56
PIK3CG P48736 1/20 0.56
GSK3B P49841 1/20 0.56
CAMKK2 Q96RR4 1/20 0.56
CAMK2D Q13557 3/20 0.55
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
AURKA O14965 1/20 0.51
PDGFRB P09619 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8837776 0.91 ABL1 (0.70) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL3509891 0.90 ABL1 (0.74) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL8837875 0.87 ABL1 (0.78) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL8837783 0.86 CSNK2A1 (0.67) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL8837795 0.86 ABL1 (0.80) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL1255 0.86 ABL1 (0.80) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL8837864 0.86 ABL1 (0.62) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL3511762 0.85 ABL1 (0.73) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL8837903 0.85 PRKCA (0.83) ABL1BCRPRKCACSNK2A1SRC
SCHEMBL8837857 0.85 ABL1 (0.76) ABL1BCRPRKCACSNK2A1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5612340-A ANTITUMOR AGENTS CIBA-GEIGY CORPORATION (US) 1997-03-18 US claimed
US-5612340-A ANTITUMOR AGENTS CIBA-GEIGY CORPORATION (US) 1997-03-18 US disclosed