SCHEMBL8839151

SCHEMBL8839151

C=CCOC(=O)c1ccc(N(C(=O)CF)c2ccc3c(c2)C(C)(C)CCC3(C)C)cc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RXRA P19793 13/20 0.46
RXRB P28702 13/20 0.46
RXRG P48443 13/20 0.46
RARB P10826 4/20 0.41
RARG P13631 4/20 0.41
RARA P10276 3/20 0.41
CYP3A4 P08684 3/20 0.40
CYP26B1 Q9NR63 1/20 0.39
CYP26A1 O43174 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8839144 0.91 RXRA (0.47) RXRARXRBRXRGRARBRARG
SCHEMBL8839361 0.89 RXRA (0.48) RXRARXRBRXRGRARBRARG
SCHEMBL8100597 0.88 RXRA (0.44) RXRARXRBRXRGRARBRARG
SCHEMBL8100803 0.88 RXRA (0.44) RXRARXRBRXRGRARBRARG
SCHEMBL7876781 0.84 RXRA (0.44) RXRARXRBRXRGRARBRARG
SCHEMBL8102470 0.82 RXRA (0.43) RXRARXRBRXRGRARBRARG
SCHEMBL5084705 0.81 RXRA (0.64) RXRARXRBRXRGRARBRARG
SCHEMBL8749101 0.80 RXRA (0.41) RXRARXRBRXRGRARBRARG
SCHEMBL7885957 0.80 RXRA (0.42) RXRARXRBRXRGRARBRARG
SCHEMBL8839082 0.78 CYP26B1 (0.46) RXRARXRBRXRGRARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688817-A SKIN DISORDERS, ANTIINFLAMMATORY AGENTS, IMMUNOLOGY AND RHEUMATIC DISORDERS CENTRE INT'L. DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 1997-11-18 US disclosed
US-5668156-A TREATMENT OF WARTS, ACNE, PSORIASIS, CORNEOPATHIES, KETONES CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (CIRD GALDERMA) (FR) 1997-09-16 US disclosed
US-5597839-A TREATMENT OF SKIN DISORDERS OR ANTIINFLAMMATORY AGENTS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (CIRD GALDERMA) (FR) 1997-01-28 US disclosed
US-5567721-A AROMATIC UREA COMPOUND FOR SKIN DISORDER, RHEUMATIC DISEASE, RESPIRATORY DISORDER AND EYE DISORDER CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (FR) 1996-10-22 US disclosed
US-5439925-A Skin disorders, rheumatic diseases CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (CIRD GALDERMA) (FR) 1995-08-08 US disclosed
US-5387594-A Administering for topical and systemic treatment of CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (CIRD GALDERMA) (FR) 1995-02-07 US disclosed