SCHEMBL8840423

SCHEMBL8840423

CCCCOc1ccc([C@H]2CC[C@@H](N(OCc3ccccc3)c3ccnc(COC)c3OC)CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.36
CYP2C9 P11712 3/20 0.34
CYP3A4 P08684 1/20 0.34
KCNH2 Q12809 1/20 0.34
RAB9A P51151 1/20 0.33
TP53 P04637 1/20 0.33
RORC P51449 1/20 0.33
S1PR1 P21453 1/20 0.33
KDM1A O60341 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.32
SPHK1 Q9NYA1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8840399 0.97 HRH3 (0.35) HRH3CYP2C9CYP3A4KCNH2S1PR1
SCHEMBL8840454 0.93 TP53 (0.34) HRH3TP53KDM1AMAOAMAOB
SCHEMBL8840408 0.92 FOXM1 (0.34) HRH3CYP2C9CYP3A4KCNH2RAB9A
SCHEMBL8840410 0.92 FOXM1 (0.34) HRH3CYP2C9CYP3A4KCNH2RAB9A
SCHEMBL8840417 0.90 GRM2 (0.34)
SCHEMBL8840437 0.88 KDM1A (0.31) HRH3KDM1AMAOAMAOBMRGPRX4
SCHEMBL8840554 0.88 MAPT (0.33) CYP3A4TP53RORCKDM1AMAOA
SCHEMBL8840395 0.87 LRRK2 (0.31)
SCHEMBL9035774 0.86 KDM4E (0.35) HRH3KDM1AMAOAMAOBMRGPRX4
SCHEMBL8840416 0.82 TP53 (0.35) HRH3CYP2C9CYP3A4KCNH2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650417-A Substituted pyridines, their preparation, and their use as pesticides and fungicides HOECHST SCHERING AGREVO GMBH (DE) 1997-07-22 US disclosed
EP-0719255-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES Hoechst Schering AgrEvo GmbH (DE) 1996-07-03 EP disclosed
WO-1995007890-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES HOECHST SCHERING AGREVO GMBH (DE) 1995-03-23 WO disclosed