SCHEMBL8840554

SCHEMBL8840554

COCc1nccc(N(OCc2ccccc2)[C@H]2CC[C@@H](c3ccc(OC(C)C)cc3)CC2)c1OC

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.33
THRB P10828 2/20 0.33
RORC P51449 1/20 0.31
KDM1A O60341 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
TSHR P16473 1/20 0.30
MRGPRX4 Q96LA9 1/20 0.30
MCL1 Q07820 1/20 0.30
GMNN O75496 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
DRD2 P14416 1/20 0.30
HPGD P15428 1/20 0.30
DRD4 P21917 1/20 0.30
DRD3 P35462 1/20 0.30
PMP22 Q01453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8840395 0.93 LRRK2 (0.31)
SCHEMBL8840417 0.90 GRM2 (0.34)
SCHEMBL8840454 0.90 TP53 (0.34) MAPTKDM1AMAOAMAOBMRGPRX4
SCHEMBL8840437 0.88 KDM1A (0.31) KDM1AMAOAMAOBMRGPRX4
SCHEMBL8840399 0.88 HRH3 (0.35) KDM1AMAOAMAOBMRGPRX4CYP3A4
SCHEMBL8840410 0.86 FOXM1 (0.34) KDM1AMAOAMAOBMRGPRX4TP53
SCHEMBL8840408 0.86 FOXM1 (0.34) KDM1AMAOAMAOBMRGPRX4TP53
SCHEMBL9035774 0.84 KDM4E (0.35) KDM1AMAOAMAOBTSHRMRGPRX4
SCHEMBL8840430 0.80 KMT2A (0.33) ALDH1A1
SCHEMBL8840443 0.80 L3MBTL1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650417-A Substituted pyridines, their preparation, and their use as pesticides and fungicides HOECHST SCHERING AGREVO GMBH (DE) 1997-07-22 US disclosed
EP-0719255-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES Hoechst Schering AgrEvo GmbH (DE) 1996-07-03 EP disclosed
WO-1995007890-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES HOECHST SCHERING AGREVO GMBH (DE) 1995-03-23 WO disclosed