SCHEMBL8842852

SCHEMBL8842852

CCOC(=O)CC(C)N1CC(=O)N(Cc2ccccc2)c2ccc(C#CSCCNC(=O)OC(C)(C)C)cc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.38
ITGA2B P08514 10/20 0.38
IDO1 P14902 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
MAPT P10636 2/20 0.32
PKM P14618 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SIGMAR1 Q99720 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7326612 0.89 ITGB3 (0.38) ITGB3ITGA2BSIGMAR1
SCHEMBL7334965 0.86 ITGB3 (0.38) ITGB3ITGA2BHDAC1HDAC6MAPT
SCHEMBL7327168 0.84 SIGMAR1 (0.37) ITGB3ITGA2BHDAC1HDAC6PDCD1
SCHEMBL7329988 0.82 ADORA3 (0.36) ITGB3ITGA2BSIGMAR1
SCHEMBL7324001 0.81 ITGB3 (0.39) ITGB3ITGA2BHDAC1HDAC6MAPT
SCHEMBL7324841 0.79 ITGB3 (0.44) ITGB3ITGA2BMAPTALDH1A1
SCHEMBL7331886 0.79 ITGB3 (0.33) ITGB3ITGA2BHDAC1HDAC6MAPT
SCHEMBL7334527 0.79 ITGB3 (0.35) ITGB3ITGA2B
SCHEMBL7328359 0.79 ITGB3 (0.43) ITGB3ITGA2BMAPTPKMALDH1A1
SCHEMBL7321894 0.78 ITGB3 (0.35) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663166-A ANTICOAGULANTS OF 1,4-BENZODIAZEPINE-2,5-DIONE AND 2-BENZOAZEPINE-1,4-DIONE DERIVATIVES; PREVENTS FIBRINOGEN BINDING NECESSARY FOR PLATELET AGGREGATION; SIDE EFFECT REDUCTION, E.G. EXCESSIVE BLEEDING GENENTECH, INC. (US) 1997-09-02 US disclosed