SCHEMBL8844387

SCHEMBL8844387

COC(=O)/C=C(/C(=O)OC)C(C)Br

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28826497 0.85 ALDH1A1 (0.33) HCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL27714989 0.83 HCAR2 (0.40) HCAR2KEAP1NFE2L2ALDH1A1
Hydrochloric Acid SCHEMBL27910123 0.81 HCAR2 (0.39) HCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL3161004 0.79 HCAR2 (0.37) HCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL6432413 0.74 HCAR2 (0.40) HCAR2KEAP1NFE2L2
SCHEMBL6432409 0.74 HCAR2 (0.40) HCAR2KEAP1NFE2L2
SCHEMBL6432420 0.74 HCAR2 (0.40) HCAR2KEAP1NFE2L2
SCHEMBL16732163 0.72 ADAM17 (0.31) HCAR2KEAP1NFE2L2
SCHEMBL7771274 0.70 HCAR2 (0.46) HCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL5953576 0.70 HCAR2 (0.46) HCAR2KEAP1NFE2L2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5627170-A Phosphonic acid compound containing heterocyclic substituents, pharmaceutical composition contains same and a method of treating calcium metabolism disturbance BOEHRINGER MANNHEIM GMBH (DE) 1997-05-06 US disclosed
US-5538957-A OSTEOPOROSIS BOEHRINGER MANNHEIM GMBH (DE) 1996-07-23 US disclosed