SCHEMBL884449

SCHEMBL884449

CC(C)Cc1ccc(-c2cc(F)ccc2C(Cc2cccnc2)c2cccnc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 8/20 0.44
KCNH2 Q12809 6/20 0.44
GRM2 Q14416 2/20 0.42
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.38
TBXAS1 P24557 2/20 0.37
ADRB3 P13945 2/20 0.37
ADRB1 P08588 1/20 0.37
ALOX5AP P20292 1/20 0.37
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5038360 0.91 KCNA5 (0.48) KCNA5KCNH2GRM2ALDH1A1CYP3A4
SCHEMBL884639 0.89 KCNA5 (0.45) KCNA5KCNH2GRM2ALDH1A1CYP3A4
SCHEMBL5033715 0.88 KCNA5 (0.50) KCNA5KCNH2GRM2ALDH1A1CYP3A4
SCHEMBL5032466 0.87 KCNA5 (0.45) KCNA5KCNH2GRM2ALDH1A1
SCHEMBL884569 0.87 KCNA5 (0.51) KCNA5KCNH2GRM2ALDH1A1
SCHEMBL885069 0.85 KCNA5 (0.56) KCNA5KCNH2GRM2ALDH1A1CYP3A4
SCHEMBL2063347 0.84 KCNA5 (0.62) KCNA5KCNH2GRM2ADRB3ADRB1
SCHEMBL884457 0.83 KCNA5 (0.51) KCNA5KCNH2ALDH1A1CYP3A4
SCHEMBL884595 0.83 KCNA5 (0.45) KCNA5KCNH2GRM2ALDH1A1
SCHEMBL884718 0.81 KCNA5 (0.51) KCNA5KCNH2GRM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940406-A2 POTASSIUM CHANNEL INHIBITORS Merck and Co., Inc. (US) 2008-07-09 EP claimed
WO-2007050348-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-05-03 WO claimed