SCHEMBL884569

SCHEMBL884569

Fc1ccc(C(Cc2cccnc2)c2cccnc2)c(-c2cccnc2)c1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 8/20 0.51
KCNH2 Q12809 6/20 0.51
CYP11B2 P19099 3/20 0.47
CYP11B1 P15538 2/20 0.47
TDO2 P48775 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GRM2 Q14416 2/20 0.40
CLK1 P49759 1/20 0.40
DYRK1A Q13627 1/20 0.40
PDE5A O76074 3/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5038360 0.93 KCNA5 (0.48) KCNA5KCNH2CYP11B2CYP11B1ALDH1A1
SCHEMBL5033715 0.92 KCNA5 (0.50) KCNA5KCNH2CYP11B2CYP11B1ALDH1A1
SCHEMBL5030913 0.89 KCNA5 (0.51) KCNA5KCNH2CYP11B2CYP11B1
SCHEMBL884457 0.89 KCNA5 (0.51) KCNA5KCNH2CYP11B2CYP11B1ALDH1A1
SCHEMBL5032466 0.89 KCNA5 (0.45) KCNA5KCNH2CYP11B2CYP11B1ALDH1A1
SCHEMBL884639 0.89 KCNA5 (0.45) KCNA5KCNH2CYP11B2CYP11B1ALDH1A1
SCHEMBL884595 0.89 KCNA5 (0.45) KCNA5KCNH2CYP11B2CYP11B1ALDH1A1
SCHEMBL884449 0.87 KCNA5 (0.44) KCNA5KCNH2ALDH1A1GRM2
SCHEMBL885069 0.87 KCNA5 (0.56) KCNA5KCNH2CYP11B2CYP11B1ALDH1A1
SCHEMBL884656 0.86 KCNA5 (0.53) KCNA5KCNH2CYP11B2CYP11B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940406-A2 POTASSIUM CHANNEL INHIBITORS Merck and Co., Inc. (US) 2008-07-09 EP claimed
WO-2007050348-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-05-03 WO claimed