SCHEMBL884457

SCHEMBL884457

Cc1cccc(-c2cc(F)ccc2C(Cc2cccnc2)c2cccnc2)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 12/20 0.51
KCNH2 Q12809 6/20 0.51
ALDH1A1 P00352 1/20 0.41
RPS6KA3 P51812 1/20 0.38
GRIN1 Q05586 2/20 0.38
GRIN2B Q13224 2/20 0.38
CYP11B2 P19099 2/20 0.38
CYP11B1 P15538 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL884639 0.89 KCNA5 (0.45) KCNA5KCNH2ALDH1A1GRIN1GRIN2B
SCHEMBL884569 0.89 KCNA5 (0.51) KCNA5KCNH2ALDH1A1CYP11B2CYP11B1
SCHEMBL5030913 0.87 KCNA5 (0.51) KCNA5KCNH2GRIN1GRIN2BCYP11B2
SCHEMBL884656 0.87 KCNA5 (0.53) KCNA5KCNH2ALDH1A1RPS6KA3CYP11B2
SCHEMBL5038360 0.87 KCNA5 (0.48) KCNA5KCNH2ALDH1A1GRIN1GRIN2B
SCHEMBL5033715 0.85 KCNA5 (0.50) KCNA5KCNH2ALDH1A1CYP11B2CYP11B1
SCHEMBL884718 0.84 KCNA5 (0.51) KCNA5KCNH2ALDH1A1CYP11B2CYP11B1
SCHEMBL884449 0.83 KCNA5 (0.44) KCNA5KCNH2ALDH1A1CYP3A4
SCHEMBL884595 0.83 KCNA5 (0.45) KCNA5KCNH2ALDH1A1CYP11B2CYP11B1
SCHEMBL5032466 0.83 KCNA5 (0.45) KCNA5KCNH2ALDH1A1CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940406-A2 POTASSIUM CHANNEL INHIBITORS Merck and Co., Inc. (US) 2008-07-09 EP claimed
WO-2007050348-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-05-03 WO claimed