SCHEMBL8844573

SCHEMBL8844573

c1ccc(CN2CCC(c3cccnc3)C2)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.59
MDM2 Q00987 1/20 0.59
TRPV6 Q9H1D0 3/20 0.56
CCR5 P51681 1/20 0.53
SIGMAR1 Q99720 1/20 0.52
PDCD1LG2 Q9BQ51 1/20 0.52
CD274 Q9NZQ7 1/20 0.52
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
DRD2 P14416 1/20 0.50
CHRNB2 P17787 1/20 0.49
CHRNA4 P43681 1/20 0.49
ROCK2 O75116 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2569983 0.93 TRPV6 (0.64) TP53MDM2TRPV6CCR5SIGMAR1
SCHEMBL6023725 0.85 MEN1 (0.68) TP53CCR5SIGMAR1MEN1KMT2A
SCHEMBL22755777 0.85 MEN1 (0.68) TP53CCR5SIGMAR1MEN1KMT2A
SCHEMBL3598146 0.85 MEN1 (0.68) TP53CCR5SIGMAR1MEN1KMT2A
SCHEMBL6956567 0.84 TP53 (0.54) TP53MDM2TRPV6CCR5SIGMAR1
SCHEMBL31328408 0.84 DRD4 (0.48) TP53MDM2TRPV6CCR5MEN1
SCHEMBL29832299 0.84 TRPV6 (0.64) TRPV6CCR5SIGMAR1MEN1KMT2A
SCHEMBL8844231 0.84 TRPV6 (0.57) TRPV6CCR5SIGMAR1MEN1KMT2A
SCHEMBL15732590 0.81 MGLL (0.46) TP53MDM2TRPV6CCR5PDCD1LG2
SCHEMBL25272839 0.81 CNR2 (0.60) TP53MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622966-A BACTERICIDES TREATING INFECTIONS WARNER-LAMBERT COMPANY (US) 1997-04-22 US disclosed
US-5446044-A Bactericides WARNER-LAMBERT COMPANY (US) 1995-08-29 US disclosed
US-5384407-A Pyrrolidine compounds WARNER-LAMBERT COMPANY (US) 1995-01-24 US disclosed
US-5342844-A 7-substituted quinolones and naphthyridones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1994-08-30 US disclosed
WO-1993016077-A1 7-SUBSTITUTED QUINOLONES AND NAPHTHYRIDONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1993-08-19 WO disclosed
US-5221676-A 7-substituted quinolones and naphthyridones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1993-06-22 US disclosed