SCHEMBL8845595

SCHEMBL8845595

COC(=O)[C@]1(NC(=O)OC(C)(C)C)CCc2cccc(Oc3ccsc3C(=O)OCc3ccccc3)c2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 2/20 0.39
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
ACHE P22303 2/20 0.37
SYK P43405 1/20 0.34
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
KLK5 Q9Y337 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CACNA1B Q00975 1/20 0.32
CTSL P07711 1/20 0.31
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
ADORA2B P29275 1/20 0.31
TACR1 P25103 1/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566163 0.89 GHSR (0.37) GHSRCA1CA2ACHESYK
SCHEMBL8520678 0.89 GHSR (0.37) GHSRCA1CA2ACHESYK
SCHEMBL8845070 0.88 GHSR (0.40) GHSRRAB9AKMT2A
SCHEMBL8844907 0.88 GHSR (0.40) GHSRRAB9AKMT2A
SCHEMBL8845267 0.82 GHSR (0.42) GHSRCA1CA2ACHESYK
SCHEMBL8845155 0.82 GHSR (0.42) GHSRCA1CA2ACHESYK
SCHEMBL8581093 0.77 GHSR (0.40) GHSRCA1CA2ACHESYK
SCHEMBL8845144 0.77 GHSR (0.39) GHSRCA1CA2ACHESYK
SCHEMBL8567143 0.76 CA1 (0.39) GHSRCA1CA2ACHESYK
SCHEMBL8575729 0.76 CA1 (0.39) GHSRCA1CA2ACHESYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5644024-A MIMICS OF PEPTIDE DOMAINS, SEQUENCE DETERMINATION, DRUGS HOFFMANN-LA ROCHE INC. (US) 1997-07-01 US disclosed