SCHEMBL8575729

SCHEMBL8575729

COC(=O)O[C@@]1(NC(=O)OC(C)(C)C)CCc2cccc(Oc3ccccc3C(=O)OCc3ccccc3)c2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
ACHE P22303 2/20 0.39
SYK P43405 1/20 0.38
ALDH1A1 P00352 2/20 0.36
GHSR Q92847 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
KLK7 P49862 2/20 0.34
KLK5 Q9Y337 2/20 0.34
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSL P07711 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567143 1.00 CA1 (0.39) CA1CA2ACHESYKALDH1A1
SCHEMBL8561422 0.90 CTSV (0.36) CA1CA2ACHEALDH1A1MAPT
SCHEMBL8573147 0.89 CYP3A4 (0.37) ALDH1A1GHSRCYP3A4TSHRMAPT
SCHEMBL8560808 0.88 SYK (0.35) CA1CA2ACHESYKALDH1A1
SCHEMBL8845267 0.87 GHSR (0.42) CA1CA2ACHESYKALDH1A1
SCHEMBL8845155 0.87 GHSR (0.42) CA1CA2ACHESYKALDH1A1
SCHEMBL8997600 0.87 SYK (0.40) CA1CA2ACHESYKALDH1A1
SCHEMBL8574453 0.87 CA1 (0.35) CA1CA2ACHESYKALDH1A1
SCHEMBL8997648 0.86 SYK (0.38) CA1CA2ACHESYKGHSR
SCHEMBL8563393 0.84 CYP3A4 (0.38) ALDH1A1GHSRCYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640618-B1 Tetrahydronaphthalene-peptide derivatives HOFFMANN LA ROCHE (CH) 1999-10-20 EP disclosed
EP-0640618-A1 Tetrahydronaphthalene-peptide derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-03-01 EP disclosed