SCHEMBL884656

SCHEMBL884656

COc1cccc(-c2cc(F)ccc2C(Cc2cccnc2)c2cccnc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 6/20 0.53
KCNH2 Q12809 5/20 0.48
CYP1A2 P05177 5/20 0.46
CYP3A4 P08684 5/20 0.46
CYP2D6 P10635 5/20 0.46
CYP2C19 P33261 5/20 0.46
CLK4 Q9HAZ1 4/20 0.46
HSD17B10 Q99714 3/20 0.46
ALOX15 P16050 2/20 0.46
PDE4B Q07343 2/20 0.43
DGAT2 Q96PD7 2/20 0.42
LMNA P02545 3/20 0.42
TSHR P16473 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPK1 P28482 2/20 0.42
NPC1 O15118 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
TP53 P04637 1/20 0.42
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL884457 0.87 KCNA5 (0.51) KCNA5KCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL884569 0.86 KCNA5 (0.51) KCNA5KCNH2ALDH1A1CYP11B1CYP11B2
SCHEMBL5030913 0.85 KCNA5 (0.51) KCNA5KCNH2CLK4PDE4BLMNA
SCHEMBL885203 0.84 KCNA5 (0.42) KCNA5KCNH2ALDH1A1CYP11B1CYP11B2
SCHEMBL5038360 0.84 KCNA5 (0.48) KCNA5KCNH2CYP3A4CYP2D6CYP2C19
SCHEMBL2064429 0.83 KCNA5 (0.69) KCNA5KCNH2DGAT2RPS6KA3
SCHEMBL5033715 0.83 KCNA5 (0.50) KCNA5KCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL884817 0.82 PDE4A (0.46) KCNA5KCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL884639 0.82 KCNA5 (0.45) KCNA5KCNH2CYP3A4HSD17B10LMNA
SCHEMBL884449 0.81 KCNA5 (0.44) KCNA5KCNH2CYP3A4ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940406-A2 POTASSIUM CHANNEL INHIBITORS Merck and Co., Inc. (US) 2008-07-09 EP claimed
WO-2007050348-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-05-03 WO claimed