SCHEMBL8850865

SCHEMBL8850865

COC(=O)CCC[N]Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
LMNA P02545 2/20 0.49
KDM4E B2RXH2 1/20 0.49
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
LTA4H P09960 2/20 0.44
TSHR P16473 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
AKT1 P31749 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
PTPRC P08575 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8852249 0.90 ALDH1A1 (0.51) ALDH1A1LMNAKDM4ECA12CA7
SCHEMBL8851560 0.84 ALOX5 (0.52) ALDH1A1LTA4HSMN1; SMN2
SCHEMBL9234737 0.83 TSHR (0.55) ALDH1A1LMNAKDM4ETSHRMEN1
SCHEMBL8851629 0.81 HDAC3 (0.57) ALDH1A1LMNALTA4HTSHRSMN1; SMN2
SCHEMBL8851854 0.80 ALDH1A1 (0.50) ALDH1A1LMNAKDM4ECA12CA7
SCHEMBL162806 0.78 HDAC1 (0.62) ALDH1A1LMNAKDM4ECA12CA7
Phosphine SCHEMBL27480219 0.76 HDAC1 (0.60) ALDH1A1LMNAKDM4ECA12CA7
SCHEMBL117432 0.76 MAPT (0.61) ALDH1A1LMNAKDM4ECA12CA7
SCHEMBL9764517 0.75 MAPT (0.65) CA12CA7CA9CA14SMN1; SMN2
SCHEMBL9404041 0.75 MAPT (0.65) CA12CA7CA9CA14SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618814-A Trisubstituted pyrimido [5,4-d] pyrimidines for modulating multi-drug resistance and pharmaceutical compositions containing these compounds DR. KARL THOMAE GMBH (DE) 1997-04-08 US disclosed
EP-0645390-A1 Trisubstituted pyrimido 5,4-d pyrimidines for modulating multidrug resistance, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1995-03-29 EP disclosed