SCHEMBL8851131

SCHEMBL8851131

COC(=O)CNC1CC[N]CC1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.42
TET2 Q6N021 1/20 0.35
TSHR P16473 4/20 0.34
RECQL P46063 1/20 0.34
METAP1 P53582 1/20 0.33
HSD17B10 Q99714 3/20 0.33
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.31
POLB P06746 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
NLRP3 Q96P20 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4489302 0.89 EPHX2 (0.40) EPHX2TET2TSHRRECQLMETAP1
SCHEMBL4450020 0.86
SCHEMBL8851320 0.84 GAA (0.42) EPHX2TSHRMETAP1HSD17B10MGAM
Hydrochloric Acid SCHEMBL76321 0.84 EPHX2 (0.47) EPHX2TET2TSHRRECQLMETAP1
SCHEMBL7440501 0.82 EPHX2 (0.55) EPHX2TET2TSHRRECQLKDM4E
SCHEMBL1977433 0.82 EPHX2 (0.59) EPHX2KDM4EKMT2APOLBNPSR1
SCHEMBL9233824 0.81 EPHX2 (0.45) EPHX2TSHRKDM4EKMT2A
SCHEMBL8851815 0.81 PPM1B (0.36) EPHX2METAP1KDM4EALDH1A1POLB
SCHEMBL2411177 0.80 EPHX2 (0.62) EPHX2KDM4EALDH1A1KMT2APOLB
SCHEMBL9141301 0.80 METAP1 (0.35) METAP1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618814-A Trisubstituted pyrimido [5,4-d] pyrimidines for modulating multi-drug resistance and pharmaceutical compositions containing these compounds DR. KARL THOMAE GMBH (DE) 1997-04-08 US disclosed
EP-0645390-A1 Trisubstituted pyrimido 5,4-d pyrimidines for modulating multidrug resistance, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1995-03-29 EP disclosed