SCHEMBL8851209

SCHEMBL8851209

CN(C)C1CCN(c2nc(N3CCOCC3)c3ncnc(N4CCc5ccccc5C4)c3n2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.41
KDM4E B2RXH2 7/20 0.40
MAPT P10636 5/20 0.40
HTT P42858 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
NPSR1 Q6W5P4 3/20 0.40
NR2F2 P24468 1/20 0.40
HIF1A Q16665 1/20 0.40
PIK3CD O00329 5/20 0.40
HPGD P15428 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
AURKA O14965 1/20 0.39
AURKB Q96GD4 1/20 0.39
MAPK1 P28482 3/20 0.39
ALDH1A1 P00352 2/20 0.39
GLA P06280 2/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 2/20 0.39
S1PR2 O95136 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9235182 1.00 LMNA (0.41) LMNAKDM4EMAPTHTTMEN1
Oxalic Acid SCHEMBL9235915 0.95 LMNA (0.44) LMNAKDM4EMAPTHTTMEN1
SCHEMBL8852171 0.94 PIK3CD (0.42) KDM4EMAPTPIK3CDHPGDSMN1; SMN2
SCHEMBL8851997 0.93 PIK3CD (0.38) LMNAKDM4EMAPTHTTMEN1
SCHEMBL8851316 0.87 PIK3CD (0.36) PIK3CDMTORPIK3C2BPIK3CAPIK3CB
SCHEMBL9229772 0.87 PIK3CD (0.42) KDM4EMAPTNPSR1PIK3CDHPGD
SCHEMBL8851157 0.86 PDE10A (0.41) LMNAMAPTHTTNPSR1MTOR
SCHEMBL8851821 0.86 PIK3CD (0.35) MEN1KMT2APIK3CDMAPK1MTOR
SCHEMBL8852164 0.84 PIK3CD (0.42) KDM4EPIK3CDHPGDSMN1; SMN2MAPK1
SCHEMBL8852150 0.83 MTOR (0.39) KDM4EMAPTPIK3CDALDH1A1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618814-A Trisubstituted pyrimido [5,4-d] pyrimidines for modulating multi-drug resistance and pharmaceutical compositions containing these compounds DR. KARL THOMAE GMBH (DE) 1997-04-08 US claimed