SCHEMBL8851997

SCHEMBL8851997

CN(C)C1CCN(c2nc(N3CCOCC3)c3ncnc(N4CCc5ccccc5C4)c3n2)CC1.c1ncc2ncncc2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 5/20 0.38
LMNA P02545 4/20 0.37
EGFR P00533 1/20 0.36
KDM4E B2RXH2 6/20 0.36
HPGD P15428 3/20 0.36
ALDH1A1 P00352 3/20 0.36
GLA P06280 2/20 0.36
GAA P10253 1/20 0.36
HTT P42858 4/20 0.36
MEN1 O00255 3/20 0.36
MAPT P10636 3/20 0.36
KMT2A Q03164 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
NR2F2 P24468 1/20 0.36
HIF1A Q16665 1/20 0.36
MTOR P42345 2/20 0.35
PTK2 Q05397 1/20 0.35
TSHR P16473 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
AURKA O14965 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8851209 0.93 LMNA (0.41) PIK3CDLMNAKDM4EHPGDALDH1A1
SCHEMBL9235182 0.93 LMNA (0.41) PIK3CDLMNAKDM4EHPGDALDH1A1
Oxalic Acid SCHEMBL9235915 0.89 LMNA (0.44) PIK3CDLMNAKDM4EHPGDALDH1A1
SCHEMBL8852171 0.88 PIK3CD (0.42) PIK3CDEGFRKDM4EHPGDALDH1A1
SCHEMBL8851316 0.81 PIK3CD (0.36) PIK3CDMTOR
SCHEMBL9229772 0.81 PIK3CD (0.42) PIK3CDKDM4EHPGDALDH1A1GLA
SCHEMBL8851821 0.80 PIK3CD (0.35) PIK3CDMEN1KMT2AMTORMAPK1
SCHEMBL8851157 0.80 PDE10A (0.41) LMNAHTTMAPTNPSR1MTOR
SCHEMBL8852164 0.78 PIK3CD (0.42) PIK3CDEGFRKDM4EHPGDALDH1A1
SCHEMBL8852150 0.78 MTOR (0.39) PIK3CDKDM4EALDH1A1MAPTMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618814-A Trisubstituted pyrimido [5,4-d] pyrimidines for modulating multi-drug resistance and pharmaceutical compositions containing these compounds DR. KARL THOMAE GMBH (DE) 1997-04-08 US claimed