SCHEMBL8851595

SCHEMBL8851595

CCCN1C(=O)CN=C(c2ccccc2)c2ccccc21

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.68
GABRG2 P18507 3/20 0.68
GABRB3 P28472 3/20 0.68
GABRA5 P31644 3/20 0.68
GABRA3 P34903 3/20 0.68
GABRA2 P47869 3/20 0.68
GABRB2 P47870 3/20 0.68
CCKBR P32239 1/20 0.68
HDAC3 O15379 1/20 0.63
HDAC1 Q13547 1/20 0.63
HDAC8 Q9BY41 1/20 0.63
HDAC6 Q9UBN7 1/20 0.63
NPSR1 Q6W5P4 2/20 0.62
GAA P10253 2/20 0.62
HTT P42858 1/20 0.62
GPR55 Q9Y2T6 1/20 0.62
SMN1; SMN2 Q16637 2/20 0.60
KDM4E B2RXH2 1/20 0.60
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9380657 0.91 HDAC3 (0.69) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7541208 0.89 GABRA1 (0.68) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6985755 0.87 GABRA1 (0.65) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL5361417 0.85 OPRK1 (0.72) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL11576361 0.85 GABRA1 (0.62) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL11577126 0.84 GABRA1 (0.61) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6949881 0.83 SMN1; SMN2 (0.63) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL11575757 0.83 GABRA1 (0.60) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL23560411 0.83 GABRA1 (0.63) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL4413309 0.83 GABRA1 (0.63) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633251-A N-2,3-dihydro-1-(2-propyl)-2-oxo-5-phenyl-1h-1,4-benzodiazepines MERCK & CO., INC. (US) 1997-05-27 US disclosed