Methylglyoxal

Methylglyoxal

SCHEMBL8854583

CC(=O)C=O.CC(O)(CO)N(N)c1ccccc1C(=O)O.CC(O)(CO)N(N)c1ccccc1C(=O)O

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 11/20 0.40
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
LMNA P02545 1/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA4 P22748 2/20 0.33
CA7 P43166 2/20 0.33
CA9 Q16790 2/20 0.33
LTB4R2 Q9NPC1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylglyoxal SCHEMBL6452706 0.88 CTSD (0.38) PTPN1ALDH1A1KDM4EMAPTTDP1
Methylglyoxal SCHEMBL8854695 0.71 PTPN1 (0.41) PTPN1ALDH1A1ALOX15KDM4EPOLB
Phthalic Acid SCHEMBL28441584 0.69 ALDH1A1 (0.61) ALDH1A1ALOX15KDM4EMAPTTDP1
SCHEMBL11796141 0.68 ALDH1A1 (0.48) PTPN1ALDH1A1ALOX15KDM4EMAPT
SCHEMBL14893324 0.67 ALDH1A1 (0.56) PTPN1ALDH1A1ALOX15KDM4EPOLB
SCHEMBL972143 0.67 ALDH1A1 (0.56) PTPN1ALDH1A1ALOX15KDM4EPOLB
Phthalic Acid SCHEMBL30288540 0.65 ALDH1A1 (0.61) ALDH1A1ALOX15KDM4EPOLBMAPT
Phthalic Acid SCHEMBL11274547 0.65 ALDH1A1 (0.61) ALDH1A1ALOX15KDM4EPOLBMAPT
Phthalic Acid SCHEMBL6551340 0.65 ALDH1A1 (0.61) ALDH1A1ALOX15KDM4EPOLBMAPT
SCHEMBL5524626 0.65 ALDH1A1 (0.48) PTPN1ALDH1A1ALOX15KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661139-A FOR INHIBITING GLYCOSYLATION OF PROTEINS TO PREVENT DISCOLORATION OF THE TEETH ALTEON INC. (US) 1997-08-26 US disclosed
WO-1996040622-A1 BIS-(2-ARYL)HYDRAZONES AS INHIBITORS OF THE FORMATION OF ADVANCED GLYCOSYLATION ENDPRODUCTS ALTEON INC. (US) 1996-12-19 WO disclosed
US-5552400-A Fused-bicyclic lactams as interleukin-1β converting enzyme inhibitors STERLING WINTHROP INC. (US) 1996-09-03 US disclosed