SCHEMBL8854822

SCHEMBL8854822

O=C1NC2C=CC=CC2=C2C1=CC(=O)c1ccccc12

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.37
CDC25B P30305 2/20 0.32
IDO1 P14902 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
AKT1 P31749 1/20 0.32
SNCA P37840 1/20 0.32
MAP2K1 Q02750 1/20 0.32
PIN1 Q13526 1/20 0.32
EHMT2 Q96KQ7 1/20 0.32
NSD1 Q96L73 1/20 0.32
EHMT1 Q9H9B1 1/20 0.32
PTPRC P08575 1/20 0.31
PTPRF P10586 1/20 0.31
PTPN1 P18031 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6163147 0.74 IDO1 (0.31) CDC25BIDO1MAOAMAOBAKT1
SCHEMBL13038795 0.67 TSHR (0.36) MAOAMAOB
SCHEMBL5904469 0.66 TNKS2 (0.36) CDC25BIDO1MAOAMAOBAKT1
SCHEMBL5531635 0.65 TNKS2 (0.36) IDO1PTPRCPTPN1
SCHEMBL3616173 0.64 MEN1 (0.34)
SCHEMBL4758533 0.63
SCHEMBL17306807 0.62 NOS2 (0.39)
SCHEMBL15624375 0.62 NOS2 (0.35)
SCHEMBL4994523 0.62
SCHEMBL13632710 0.61 GAA (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069308-B1 AZONAFIDE DERIVED TUMOR AND CANCER TARGETING COMPOUNDS GOVERNMENT OF THE UNITED STATES OF AMERICA REPRESENTED BY THE SECRETARY DEPT OF HEALTH AND HUMAN SER (US) 2017-03-29 EP disclosed
US-5703089-A ANTICANCER AGENTS KNOLL AKTIENGESELLSCHAFT (DE) 1997-12-30 US disclosed