SCHEMBL8855488

SCHEMBL8855488

O=[N+]([O-])c1nccn1C[C@H]1CO1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
CA12 O43570 5/20 0.46
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CA9 Q16790 5/20 0.46
TYMP P19971 3/20 0.45
LMNA P02545 1/20 0.45
THRB P10828 1/20 0.45
CYP2C19 P33261 1/20 0.45
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
OPRK1 P41145 1/20 0.41
TP53 P04637 1/20 0.35
HBB P68871 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NOS1 P29475 1/20 0.33
BRD4 O60885 1/20 0.32
CCR10 P46092 2/20 0.32
GRIN2B Q13224 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1614716 1.00 KMT2A (0.47) KMT2ACA12CA1CA2CA9
SCHEMBL8897393 1.00 KMT2A (0.47) KMT2ACA12CA1CA2CA9
SCHEMBL6960235 0.89 TYMP (0.41) KMT2ACA12CA1CA2CA9
SCHEMBL11390072 0.76 CA12 (0.64) KMT2ACA12CA1CA2CA9
SCHEMBL15597325 0.73 TYMP (0.56) KMT2ACA12CA1CA2CA9
SCHEMBL29579255 0.73 CA12 (0.53) KMT2ACA12CA1CA2CA9
SCHEMBL16752479 0.73 CA12 (0.53) KMT2ACA12CA1CA2CA9
SCHEMBL8530813 0.73 LMNA (0.59) KMT2ACA12CA1CA2CA9
SCHEMBL9272320 0.73 KMT2A (0.54) KMT2ACA12CA1CA2CA9
SCHEMBL10842757 0.72 KMT2A (0.41) KMT2ACA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5342959-A Process for preparing chiral [[(2-bromoethyl)-amino]methyl]-2-nitro-1H-imidazol-1-ethanol and related compounds WARNER-LAMBERT COMPANY (US) 1994-08-30 US claimed
WO-1994015922-A1 NOVEL PROCESS FOR PREPARING CHIRAL [[(2-BROMOETHYL)AMINO]METHYL]-2-NITRO-1H-IMIDAZOL-1-ETHANOL AND RELATED COMPOUNDS WARNER LAMBERT COMPANY (US) 1994-07-21 WO claimed
US-5659048-A CHEMOSENSITIZER, RADIOSENSITIZER ADMINISTERING TO PATIENTS WHOM ARE SENSITIVE TO RADIATION OR CHEMOTHERAPY BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-08-19 US disclosed
US-5652255-A ADMINISTERING NITROIMIDAZOLE DERIVATIVE NITRIC OXIDE SYNTHASE INHIBITOR; ANTITUMOR AGENTS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-07-29 US disclosed
US-5543527-A ANTITUMOR AGENTS BRITISH TECHNOLOYG GROUP LIMITED (GB) 1996-08-06 US disclosed
US-5481000-A RADIOSENSITIZERS OR CHEMOSENSITIZERS; PATENT CLAIMS CHIRAL 3-/2-HYDROXY-3-/2-NITROIMIDAZOL-1-YL/PROPYL/-2-OXAZOLIDINONE, HAVING /S/ CONFIGURATION AT OH CARBON AND FREE OF /R/ CONFIGURATION WARNER-LAMBERT COMPANY (US) 1996-01-02 US disclosed
US-5342959-A Process for preparing chiral [[(2-bromoethyl)-amino]methyl]-2-nitro-1H-imidazol-1-ethanol and related compounds WARNER-LAMBERT COMPANY (US) 1994-08-30 US disclosed