SCHEMBL8858342

SCHEMBL8858342

C1=C(/C=C/c2ccccc2)CCN(Cc2coc3ccccc23)C1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.48
DRD4 P21917 8/20 0.48
DRD3 P35462 8/20 0.48
KDM4E B2RXH2 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SIGMAR1 Q99720 2/20 0.44
HTR1A P08908 4/20 0.42
MAOB P27338 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858344 1.00 DRD2 (0.48) DRD2DRD4DRD3KDM4ESMN1; SMN2
SCHEMBL8791055 0.91 MAOA (0.45) DRD2DRD4DRD3KDM4ESMN1; SMN2
SCHEMBL8858349 0.91 MAOA (0.45) DRD2DRD4DRD3KDM4ESMN1; SMN2
SCHEMBL8790895 0.88 DRD2 (0.44) DRD2DRD4DRD3KDM4ESMN1; SMN2
SCHEMBL8790889 0.88 DRD2 (0.44) DRD2DRD4DRD3KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL8858366 0.88 DRD2 (0.43) DRD2DRD4DRD3KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL8858362 0.88 DRD2 (0.43) DRD2DRD4DRD3KDM4ESMN1; SMN2
SCHEMBL8858346 0.87 HTR1A (0.47) DRD2DRD4DRD3KDM4ESMN1; SMN2
SCHEMBL8858347 0.87 HTR1A (0.47) DRD2DRD4DRD3KDM4ESMN1; SMN2
SCHEMBL8858363 0.86 DRD2 (0.37) DRD2DRD4DRD3KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5665722-A Benzofuran derivatives as D4 receptor antagonists MERCK, SHARP & DOHME, LTD. (GB) 1997-09-09 US disclosed