SCHEMBL8858368

SCHEMBL8858368

C1=C(/C=C/c2ccc3c(c2)OCO3)CCN(Cc2coc3ccccc23)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HTR1A P08908 3/20 0.38
SIGMAR1 Q99720 2/20 0.38
CYP19A1 P11511 2/20 0.37
DRD2 P14416 3/20 0.37
DRD4 P21917 3/20 0.37
DRD3 P35462 3/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 2/20 0.37
KMT2A Q03164 2/20 0.37
USP2 O75604 1/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 3/20 0.36
CYP3A4 P08684 1/20 0.36
ATM Q13315 1/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858371 1.00 KDM4E (0.39) KDM4ESMN1; SMN2HTR1ASIGMAR1CYP19A1
SCHEMBL8858342 0.85 DRD2 (0.48) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2
SCHEMBL8858344 0.85 DRD2 (0.48) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2
SCHEMBL8858349 0.84 MAOA (0.45) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2
SCHEMBL8791055 0.84 MAOA (0.45) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2
SCHEMBL8790895 0.83 DRD2 (0.44) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2
SCHEMBL8790889 0.83 DRD2 (0.44) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2
Hydrochloric Acid SCHEMBL8858362 0.82 DRD2 (0.43) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2
Hydrochloric Acid SCHEMBL8858366 0.82 DRD2 (0.43) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2
SCHEMBL8858363 0.81 DRD2 (0.37) KDM4ESMN1; SMN2HTR1ASIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5665722-A Benzofuran derivatives as D4 receptor antagonists MERCK, SHARP & DOHME, LTD. (GB) 1997-09-09 US disclosed