SCHEMBL8858633

SCHEMBL8858633

COC(=O)C(C#N)c1cccc2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
MAPT P10636 2/20 0.44
MAPK1 P28482 2/20 0.44
HSD17B10 Q99714 2/20 0.44
CASP1 P29466 1/20 0.44
GAA P10253 2/20 0.40
LMNA P02545 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HPGD P15428 1/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
ALOX5 P09917 1/20 0.39
HIF1A Q16665 1/20 0.39
PGR P06401 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3328982 0.84 MTNR1A (0.59) MTNR1AMTNR1B
SCHEMBL27853930 0.83 ALDH1A1 (0.43) ALDH1A1MAPTGAALMNACYP1A2
SCHEMBL31724327 0.80 KMT2A (0.44) ALDH1A1KMT2AMEN1MAPTMAPK1
SCHEMBL6801211 0.80 ALDH1A1 (0.48) ALDH1A1MAPTGAALMNACYP1A2
SCHEMBL16466618 0.80 KMT2A (0.44) ALDH1A1KMT2AMEN1MAPTMAPK1
SCHEMBL28847197 0.79 ALDH1A1 (0.47) ALDH1A1KMT2AMEN1MAPK1HSD17B10
SCHEMBL1274082 0.78 KMT2A (0.43) ALDH1A1KMT2AMEN1MAPTMAPK1
SCHEMBL8721957 0.78 ALDH1A1 (0.43) ALDH1A1MAPTGAALMNACYP1A2
SCHEMBL17465785 0.78 ALDH1A1 (0.43) ALDH1A1KMT2AMEN1MAPTMAPK1
SCHEMBL16811757 0.78 CASP1 (0.49) ALDH1A1KMT2AMEN1CASP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616614-A USEFUL IN TREATMENT OF DISORDERS LINKED TO ABNORMAL MELATONIN ACTIVITY ADIR ET COMPAGNIE (FR) 1997-04-01 US disclosed
EP-0562956-B1 Naphtylalkylamines, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-09-27 EP disclosed
US-5420158-A Melatonin activity ADIR ET COMPAGNIE (FR) 1995-05-30 US disclosed
EP-0562956-A1 Naphtylalkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-09-29 EP disclosed