SCHEMBL8858734

SCHEMBL8858734

CN1CCc2nc(C3CCN(C(=O)OCc4ccccc4)CC3)sc2CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
CYP2C19 P33261 1/20 0.48
PTGDR2 Q9Y5Y4 1/20 0.45
GRIN2B Q13224 7/20 0.45
HTT P42858 1/20 0.45
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
JAK2 O60674 2/20 0.44
JAK1 P23458 2/20 0.44
TYK2 P29597 2/20 0.44
JAK3 P52333 2/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TMEM97 Q5BJF2 4/20 0.43
SIGMAR1 Q99720 4/20 0.43
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858595 0.87 SMN1; SMN2 (0.47) SMN1; SMN2NPC1RAB9ACYP2C19PTGDR2
SCHEMBL8858792 0.86 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9ACYP2C19PTGDR2
SCHEMBL8858698 0.83 SMN1; SMN2 (0.49) SMN1; SMN2NPC1RAB9ACYP2C19PTGDR2
SCHEMBL8858614 0.82 SMN1; SMN2 (0.46) SMN1; SMN2NPC1RAB9ACYP2C19PTGDR2
SCHEMBL8594128 0.78 SMN1; SMN2 (0.55) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL2710739 0.77 KMT2A (0.60) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL20135380 0.76 AADAT (0.58) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL8549063 0.75 TSHR (0.53) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL20135566 0.75 SMN1; SMN2 (0.51) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL8554012 0.75 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607944-A ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-03-04 US disclosed
EP-0639575-A1 Bicyclic heterocycles, medicaments comprising these compounds and processes for their production Dr. Karl Thomae GmbH (DE) 1995-02-22 EP disclosed