SCHEMBL8554012

SCHEMBL8554012

O=C(O)c1csc(C2CCN(C(=O)OCc3ccccc3)CC2)n1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
CYP2C19 P33261 1/20 0.54
GRIN2B Q13224 9/20 0.50
CYP2D6 P10635 4/20 0.48
CYP2C9 P11712 4/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ENPP2 Q13822 2/20 0.47
HTT P42858 1/20 0.47
JAK2 O60674 2/20 0.46
JAK1 P23458 2/20 0.46
TYK2 P29597 2/20 0.46
JAK3 P52333 2/20 0.46
FAAH O00519 1/20 0.46
CYP3A4 P08684 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3594917 0.89 SMN1; SMN2 (0.51) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL20542493 0.83 SMN1; SMN2 (0.43) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL15453812 0.82 ENPP2 (0.56) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL13910005 0.81 SCN9A (0.47) SMN1; SMN2CYP2C19CYP2C9MEN1KMT2A
SCHEMBL20541282 0.81 GPR119 (0.49) SMN1; SMN2NPC1RAB9AHTTFAAH
SCHEMBL20705254 0.81 AADAT (0.54)
SCHEMBL27035855 0.80 GRIN2B (0.66) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL8594128 0.78 SMN1; SMN2 (0.55) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL2952296 0.78 CASP8 (0.42) NPSR1HTTFAAH
SCHEMBL28306819 0.78 PTGDR2 (0.49) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817677-A ANTITHROMBOSIS AGENTS DR. KARL THOMAE GMBH (DE) 1998-10-06 US disclosed
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed