SCHEMBL8859025

SCHEMBL8859025

OCCOCCC1c2ccccc2CCc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 9/20 0.49
RET P07949 1/20 0.49
HRH1 P35367 8/20 0.42
HTR2C P28335 2/20 0.39
CHRM1 P11229 1/20 0.39
DRD2 P14416 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
CHRM3 P20309 1/20 0.39
ADRA1A P35348 1/20 0.39
DRD3 P35462 1/20 0.39
KCNH2 Q12809 1/20 0.39
ACP3 P15309 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
IDO1 P14902 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7167654 0.82 HTR2A (0.59) HTR2ARETHRH1HTR2CCHRM1
SCHEMBL8201075 0.79 HTR2A (0.55) HTR2ARETHRH1HTR2CCHRM1
SCHEMBL11229592 0.75 ALDH1A1 (0.39) HTR2ADRD2ADRA2BADRA2CADRA1A
SCHEMBL9875531 0.74 HTR2A (0.63) HTR2ARETHRH1HTR2CCHRM1
SCHEMBL8712643 0.74 RET (0.44) HTR2ARETACP3IDO1
Di(Hydroxyethyl)Ether SCHEMBL6251141 0.72 TSHR (0.50) HTR2CMEN1KMT2AIDO1
SCHEMBL11837153 0.71 HTR2A (0.46) HTR2ARETHRH1HTR2CCHRM1
SCHEMBL24631299 0.71 HTR2A (0.66) HTR2ARETHRH1HTR2C
SCHEMBL8255138 0.71 HTR2A (0.78) HTR2ARETHRH1HTR2CCHRM1
SCHEMBL11220205 0.70 ALDH1A1 (0.45) HTR2ADRD2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997022342-A1 NOVEL METHOD NOVO NORDISK A/S (DK) 1997-06-26 WO disclosed
EP-0585314-B1 NOVEL HETEROCYCLIC CARBOXYLIC ACIDS NOVO NORDISK AS (DK) 1996-09-18 EP disclosed
US-5348965-A N-substituted azaheterocyclic carboxylic acids NOVO NORDISK A/S (DK) 1994-09-20 US disclosed
EP-0585314-A1 NOVEL HETEROCYCLIC CARBOXYLIC ACIDS. NOVO NORDISK AS (DK) 1994-03-09 EP disclosed
WO-1992020658-A1 NOVEL HETEROCYCLIC CARBOXYLIC ACIDS NOVO NORDISK A/S (DK) 1992-11-26 WO disclosed