SCHEMBL8859907

SCHEMBL8859907

CC(C)C(CC(C=O)C(=O)OC(C)(C)C)C(N)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
EPHX1 P07099 3/20 0.33
LMNA P02545 1/20 0.33
ANPEP P15144 1/20 0.33
ERAP2 Q6P179 1/20 0.33
APP P05067 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
NR1H4 Q96RI1 2/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
KIF11 P52732 1/20 0.30
GRIA4 P48058 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7356998 0.73 LMNA (0.40) EPHX1LMNAANPEPERAP2AKR1C3
SCHEMBL6706683 0.67 CTSK (0.33)
SCHEMBL27679365 0.67 CTSK (0.33)
SCHEMBL11014866 0.65 KMT2A (0.50) EPHX1LMNANR1H4KIF11GRIA4
SCHEMBL16355708 0.65 TP53 (0.45) TP53TSHREPHX1ANPEPERAP2
SCHEMBL20235896 0.65 TP53 (0.45) TP53TSHREPHX1ANPEPERAP2
SCHEMBL28598195 0.64 SMN1; SMN2 (0.39) TSHRLMNAAPP
SCHEMBL27535170 0.64 CYP3A4 (0.42) LMNAAPPGRIN2DGRIN3BGRIN1
SCHEMBL5425377 0.64 CTSK (0.37) LMNA
SCHEMBL8071393 0.64 KMT2A (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5654445-A INTERMEDIATES FOR RENIN INHIBITORS, HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1997-08-05 US disclosed
US-5627182-A RENIN INHIBITORS FOR USE AS HYPOTENSIVE AGENTS CIBA GEIGY CORPORATION (US) 1997-05-06 US disclosed