SCHEMBL8860177

SCHEMBL8860177

CN1[C@@H]2CCC[C@@]1(OC(=O)C(C(=O)O)c1ccccc1)CC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.39
CYP2D6 P10635 4/20 0.38
LMNA P02545 2/20 0.38
CYP2C9 P11712 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SRC P12931 1/20 0.37
CHRM2 P08172 6/20 0.37
CHRM1 P11229 6/20 0.37
CHRM3 P20309 6/20 0.37
CHRM5 P08912 5/20 0.37
CHRM4 P08173 5/20 0.37
BLM P54132 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP3A4 P08684 2/20 0.37
CYP1A2 P05177 1/20 0.37
HTT P42858 1/20 0.36
HTR2C P28335 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5793665 0.85 CYP2D6 (0.39) SLC6A9CYP2D6LMNACYP2C9HSD17B10
SCHEMBL9640284 0.79 CHRM2 (0.46) CHRM2CHRM1CHRM3CHRM4MEN1
SCHEMBL2488210 0.78 TYR (0.41) KDM4E
SCHEMBL3485175 0.76 DRD3 (0.42) SLC6A9CYP2D6LMNACHRM2CHRM1
SCHEMBL5790059 0.76 ALDH1A1 (0.40) LMNASMN1; SMN2KDM4EPOLBKMT2A
SCHEMBL3690763 0.75 CYP1A2 (0.51) CYP2D6CYP1A2POLB
Hydrochloric Acid SCHEMBL4152474 0.75 DRD3 (0.41) CYP2D6LMNACHRM2CHRM1CHRM3
SCHEMBL18978323 0.70 SRC (0.52) CYP2D6LMNASRCCHRM2CHRM1
SCHEMBL1851579 0.69 KMT2A (0.39) KDM4EMEN1POLBKMT2AALDH1A1
Hydrochloric Acid SCHEMBL6678403 0.69 MEN1 (0.50) CYP2D6LMNACHRM2CHRM1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637601-A ANTIPERSPIRANT, MYDRIATIC, ANTISECRETORY AGENTS UNIVERSITY OF FLORIDA (US) 1997-06-10 US disclosed
US-5618826-A Anticholinergic compounds, compositions and methods of treatment UNIVERSITY OF FLORIDA (US) 1997-04-08 US disclosed
US-5610188-A MYDRIATICS, ANTIPERSPIRANTS UNIVERSITY OF FLORIDA (US) 1997-03-11 US disclosed
US-5418244-A Antiperspirants, mydriatic UNIVERSITY OF FLORIDA (US) 1995-05-23 US disclosed
US-5258388-A Antisecretory agents, mydriatic agents and antiperspirants UNIVERSITY OF FLORIDA (US) 1993-11-02 US disclosed
US-5223528-A Antisecretory agents, mydriatics, antiperspirants UNIVERSITY OF FLORIDA (US) 1993-06-29 US disclosed
EP-0238982-B1 ANTICHOLINERGIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHOD OF TREATMENT UNIVERSITY OF FLORIDA (US) 1993-03-10 EP disclosed
WO-1987005603-A1 ANTICHOLINERGIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHOD OF TREATMENT UNIVERSITY OF FLORIDA (US) 1987-09-24 WO disclosed